Alprazolam + Sertraline Pharmacology

Alprazolam + Sertraline

About Alprazolam + Sertraline
N/A
Mechanism of Action of Alprazolam + Sertraline
N/A
Pharmacokinets of Alprazolam + Sertraline
N/A
Onset of Action for Alprazolam + Sertraline
N/A
Duration of Action for Alprazolam + Sertraline
N/A
Half Life of Alprazolam + Sertraline
N/A
Side Effects of Alprazolam + Sertraline
N/A
Contra-indications of Alprazolam + Sertraline
N/A
Special Precautions while taking Alprazolam + Sertraline
N/A
Pregnancy Related Information
Contraindicated, since Alprazolam is contraindicated in pregnancy
Old Age Related Information
N/A
Breast Feeding Related Information
Contraindicated, since Alprazolam is contraindicated in pregnancy
Children Related Information
N/A
Indications for Alprazolam + Sertraline
Anxiety
Interactions for Alprazolam + Sertraline
N/A
Typical Dosage for Alprazolam + Sertraline
DOSAGE: 1 tablet / day
Varies with weight and severity of the disease. Following Alprazolam combinations are available in the market. The dosage has to be decided by the treating specialist.
Each tablet contains
Alprazolam 0.25 mg + Sertraline 25 mg or
Alprazolam 0.5 mg + Sertraline 25 mg or
Alprazolam 0.5 mg + Sertraline 50 mg
Schedule of Alprazolam + Sertraline
N/A
Storage Requirements for Alprazolam + Sertraline
N/A
Effects of Missed Dosage of Alprazolam + Sertraline
N/A
Effects of Overdose of Alprazolam + Sertraline
N/A

Alprazolam

About Alprazolam
Benzodiazepine derivative, Anti anxiety.
Mechanism of Action of Alprazolam
Alprazolam mainly acts on Limbic system and ascending reticular formation in the CNS and binds to the BZD receptor. The binding will facilitates GABA mediated chloride channel opening and produce hyperpolarisation. This will produce an increase in the concentration of the inhibitory neurotransmitter GABA and increase in chloride ions and decreases firing rate of neuron. This in turn alters normal functions of the body.
Pharmacokinets of Alprazolam
Absorption: It is well absorbed after oral administration. Distribution: It is distributed widely in the body in protein bound form. Metabolism: It is metabolised to active and inactive metabolite in the liver. Excretion: Drug is excreted in urine.
Onset of Action for Alprazolam
15 - 30 minutes
Duration of Action for Alprazolam
12 - 16 hours
Half Life of Alprazolam
12 -15 hours
Side Effects of Alprazolam
1.Ataxia
2.Drowsiness
3.Light headedness
4. Slurred speech
5.Nausea
6.Constipation or diarrhoea
7.Tremor
8.Dependence
9.Anorexia
0.Confusion
11.Light headedness
12.Mood changes
13.Muscle rigidity
14.Amnesia
Contra-indications of Alprazolam
1.Hypersensitivity to Benzodiazepines
2.Acute angle closure glaucoma
Special Precautions while taking Alprazolam
1.Renal impairment
2.Hepatic impairment
3.Pulmonary insufficiency
4.Drug abuse
5.Bipolar disorder
6.Driving vehicles and operating machines and people involving any other dangerous activities
Pregnancy Related Information
Contraindicated
Old Age Related Information
Use with caution
Breast Feeding Related Information
Contraindicated
Children Related Information
Contraindicated
NEONATES- contraindicated
Indications for Alprazolam
1.For the short-term management of anxiety,
2.Treatment of Panic disorder.
Interactions for Alprazolam
Alcohol & other CNS depressants: Enhanced CNS effects.
Aminophylline: Antagonizes the sedative effect.
Cimetidine, Oral contraceptives, Disulfiram, Fluoxetine, Isoniazid, Ketoconazole, Metoprolol, Propoxyphene, Propranolol,
Valproic Acid: Elimination of alprazolam decreased due to inhibition of hepatic metabolism leading to enhanced activity.
Digoxin: Increase in serum concentration of Digoxin.
Imipramine & Desipramine: Enhanced activity of these drugs.
Levodopa: Decrease in antiparkinsonism efficacy.
Rifampicine: Decreases efficacy.
Typical Dosage for Alprazolam
Adult:
Anxiety: 0.25 - 0.5 mg every 8 hours in a day. Depending on the severity of the disease the dose can be gradually increased every 3 or 4 days.
Maximum dose: 4 mg / day in divided dose.
Anxiety with depression: 0.5 mg every 8 hours in a day
Maintenance dose: 1.5 - 4.5 mg/ day in divided dose
Panic disorder: starting dose: 1.5 mg /day in 3 divided dose. Depending on the severity of the disease the dose can be gradually increased every 3 or 4 days.

Children: Not recommended
Schedule of Alprazolam
H
Storage Requirements for Alprazolam
The drug should be kept at 15 - 30 degree C in a tightly closed container. Keep out of the reach of children
Effects of Missed Dosage of Alprazolam
Take the missed dose as soon as noticed and if it is the time for next dose then skip the missed dose.
Effects of Overdose of Alprazolam
Give supportive measures and symptomatic treatment. Flumazenil can be given as antagonist. Hypotension can be treated with vasopressors.If the patient is conscious induce emesis followed by charcoal administration

Sertraline

About Sertraline
Selective Serotonin Reuptake Inhibitor (SSRI), Antidepressant, Antidepressant
Mechanism of Action of Sertraline
Sertraline blocks the re-uptake of neurotransmitter Serotonin from the synapse in to the presynaptic nerve terminal in the CNS. This will prolong the action of Serotonin (5HT) and it is useful in the treatment of depression.
Pharmacokinets of Sertraline
Absorption: Sertraline is well absorbed after oral administration.
Distribution: It is distributed in the body in protein bound form.
Metabolism: It undergoes hepatic metabolism and produces active metabolites.
Excretion: Excreted in urine and faeces.
Onset of Action for Sertraline
1 week
Duration of Action for Sertraline
N/A
Half Life of Sertraline
26 hours
Side Effects of Sertraline
1. Insomnia
2. Nausea
3. Diarrhoea
4. Headache
5. Fatigue
6. Dizziness
7. Tremor
8. Somnolence
9. Dry mouth
10. Anorexia
11. Impotence
12. Increased sweating
13. Constipation
14. Dyspepsia
15. Agitation
16. Malaise
17. Abdominal pain












Contra-indications of Sertraline
1. Hypersensitivity to Sertraline
2. Patient on MAOI (Monoamine oxidase inhibitor) therapy
Special Precautions while taking Sertraline
1. Hepatic impairment
2. Renal impairment
3. Epilepsy
4. Hypomania
5. Metabolic disorder
6. Alcoholics
7. Patient on MAOI therapy (Discontinue the MAO inhibitor at least 2 weeks before Sertraline is started)
8. Use cautiously in patient at risk for suicide
9. Use caution while driving vehicle, operating machine and activities requiring mental alertness or judgment
Pregnancy Related Information
Use with caution
Old Age Related Information
Use with caution
Breast Feeding Related Information
Use with caution
Children Related Information
Contraindicated
NEONATES: Contraindicated

Indications for Sertraline
1. Panic disorder
2. Post traumatic stress disorder
3. Depression
4. Obsessive compulsive disorder
Interactions for Sertraline
Desipramine, diazepam, digoxin and alcohol : No significant interaction reported.
Lithium: On concomitant use, increased incidence of mild to moderate tremors has been observed.
Warfarin : Sertraline with warfarin may increase prothrombin time.
Typical Dosage for Sertraline
Adult
Panic disorder, Post traumatic stress disorder: Initial dose: 25 mg / day dose can be gradually increased every week if sufficient response does not occurs.
Maximum dose: 200 mg / day
Depression, Obsessive compulsive disorder: Initial dose: 50 mg / day dose can be gradually increased every week if sufficient response does not occur.
Maximum dose: 200 mg / day

Schedule of Sertraline
H
Storage Requirements for Sertraline
Store at 15 - 30 degree C in a tightly closed container. Protect from direct light and heat. Keep out of the reach of children.
Effects of Missed Dosage of Sertraline
Take the missed dose as soon as noticed and if it is the time for next dose then skip the missed dose.
Effects of Overdose of Sertraline
Give supportive measures and symptomatic treatment. Activated charcoal can be given to reduce the absorption of the drug.

Home Delivery for Alprazolam + Sertraline in Your City

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Alprazolam + Sertraline is a generic medicine name and there are several brands available for it. Some of the brands for alprazolam + sertraline might be better known than alprazolam + sertraline itself. If the pharmacy that's willing to deliver medicines to your home doesn't have alprazolam + sertraline in stock, you can ask for one of the branded alternatives for alprazolam + sertraline.