Ceftriaxone + Vancomycin Pharmacology

Ceftriaxone + Vancomycin

About Ceftriaxone + Vancomycin
N/A
Mechanism of Action of Ceftriaxone + Vancomycin
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Pharmacokinets of Ceftriaxone + Vancomycin
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Onset of Action for Ceftriaxone + Vancomycin
N/A
Duration of Action for Ceftriaxone + Vancomycin
N/A
Half Life of Ceftriaxone + Vancomycin
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Side Effects of Ceftriaxone + Vancomycin
N/A
Contra-indications of Ceftriaxone + Vancomycin
N/A
Special Precautions while taking Ceftriaxone + Vancomycin
N/A
Pregnancy Related Information
Use with caution
Old Age Related Information
Use with caution
Breast Feeding Related Information
Use with caution
Children Related Information
Use with caution
Indications for Ceftriaxone + Vancomycin
1.Bacterial meningitis
2.Prophylaxis of shunt infections
3.Brain abscess
4.Suppurative intracranial infections
5.Abdominal infections
6.Pneumonia
7.Acute bacterial endocarditis.
8.Bone and joint infections
9.Over whelming post-splenectomy sepsis
10.Purpura fulminans
Interactions for Ceftriaxone + Vancomycin
N/A
Typical Dosage for Ceftriaxone + Vancomycin
(Ceftriaxone-Vancomycin) can be administrated through slow intravenous injection over atleast 60 minutes. Do not dilute with calcium containing solutions .

Doses: Adults: (Ceftraixone 2 g + Vancomycin 1 g ) 3g b.i.d

Paediatric Doses : 60mg / kg body weight

Doses should be adjusted in patients with marked decrease in the renal function
Schedule of Ceftriaxone + Vancomycin
N/A
Storage Requirements for Ceftriaxone + Vancomycin
N/A
Effects of Missed Dosage of Ceftriaxone + Vancomycin
N/A
Effects of Overdose of Ceftriaxone + Vancomycin
N/A

Ceftriaxone

About Ceftriaxone
Third Generation Cephalosporin antibiotic(Parenteral).
Mechanism of Action of Ceftriaxone
Ceftriaxone is a 3rd generation cephalosporin which exerts its bactericidal action against both gram positive & gram negative organisms by inhibiting bacterial cell wall synthesis. Ceftriaxone inhibits transpeptidase & thus prevents cross linking of bacterial cell wall. Transpeptidase & associated proteins constitute various types of specific binding proteins which have affinity for cephalosporins like Ceftriaxone.

Pharmacokinets of Ceftriaxone
Absorption: Orally not well absorbed & should be given parenterally, Distribution: widely distributed & good CSF penetration, Metabolism: A portion of the drug is metabolized in the body. Excretion:
Excreted through urine & bile. A small portion of drug appears in breast milk.
Onset of Action for Ceftriaxone
Sudden
Duration of Action for Ceftriaxone
8 hours
Half Life of Ceftriaxone
N/A
Side Effects of Ceftriaxone
1.Nausea
2.Vomiting
3.Diarrhoea
4.Superinfection
5.Skin rash
6.Urticaria
7.Pseudomembranous colitis
8.Pain at site of injection
Contra-indications of Ceftriaxone
Hypersensitivity to Ceftriaxone
Special Precautions while taking Ceftriaxone
1.Hepatic impairment
2.Renal impairment
Pregnancy Related Information
Use with caution
Old Age Related Information
May be used
Breast Feeding Related Information
Use with caution
Children Related Information
May be used
Neonates: Use with caution
Indications for Ceftriaxone
1.Meningitis
2.Septicaemia
3.Typhoid
4.UTI
5.Prophylaxis in surgical infections
6.Lower respiratory tract infections
7.Pneumonia
8.Pelvic inflammatory disease
9.STD
10.Bacteraemia
Interactions for Ceftriaxone
Alcohol: Disulfiram like reaction.
Aminoglycosides & fruesmide: Nephrotoxicity potentiated.
Chloramphenicol: Decreased efficacy of ceftriaxone.
Typical Dosage for Ceftriaxone
Adults: 1g to 2gm I.M. or I.V. Once daily or two times daily
Maximum adult dose: Up to 4gm/day
Meningitis & Endocarditis: 1 to 2gm I.M. or I.V twice daily; two weeks for meningitis & four weeks for endocarditis
Gonorrhea: 250mg once daily

Children: 50 to 100 mg/kg/day I.M or I.V. two times daily
Maximum child dose: 2g/day
Meningitis & Endocarditis: 50 to 100 mg/kg/day twice daily; two weeks for meningitis & four weeks for endocarditis

Schedule of Ceftriaxone
H
Storage Requirements for Ceftriaxone
N/A
Effects of Missed Dosage of Ceftriaxone
Take the missed dose as soon as noticed and if it is the time for next dose then skip the missed dose. Continue the regular schedule. Do not double the dose.
Effects of Overdose of Ceftriaxone
Symptoms of over dosage include neuromuscular disorders & some times seizure may get precipitated. Treatment is supportive.

Vancomycin

About Vancomycin
A tricyclic glycopeptide antibiotic.
Mechanism of Action of Vancomycin
Vancomycin binds to the terminal dipeptide sequence of peptidoglycan and inhibits the association and cross linking of peptidoglycan and as the result inhibit cell wall synthesis.
Pharmacokinets of Vancomycin
Absorption: It is well absorbed after parenteral administration.
Distribution: It is very widely distributed in the body.
Excretion: It is excreted through urine.
Onset of Action for Vancomycin
Within minute
Duration of Action for Vancomycin
6 - 8 hours
Half Life of Vancomycin
4 - 6 hours
Side Effects of Vancomycin
1. Thrombophlebitis
2. Pain at the site of injection
3. Fever
4. Necrosis
5. Chills
6. Urticaria
7. Rashes
8. Flushing
9. Neutropenia
10. Oototoxicity
Contra-indications of Vancomycin
1.Hypersensitive to Vancomycin
Special Precautions while taking Vancomycin
1. Renal impairment
2. Hepatic dysfunction
3. Hearing problems
Pregnancy Related Information
Use with caution
Old Age Related Information
Use with caution
Breast Feeding Related Information
Use with caution
Children Related Information
Use with caution
NEONATES: Use with caution
Indications for Vancomycin
1. Endocarditis
2. Pseudomembranous enterocolitis
3. Methicillin resistant Staphylococcus aureus infection
4. Staphylococcal enterocolitis
Interactions for Vancomycin
Anion-exchange resins: Antagonism of oral vancomycin by cholestyramine.
Aminoglycosides: Risk of nephrotoxicity may be increased.
Anaesthetics: Erythema and histamine like flushing in children.
Nondepolorizing Muscle Relaxants: The neuromuscular blockade may be enhanced.

Typical Dosage for Vancomycin
Adult (IV dose):500 mg every four times a day
Enterocolitis (oral) 0.5 - 2 g / day in four divided dose for 10 days
Children :( IV dose) 40 mg /kg body weight / day in four divided dose
Neonates: Initial dose: 15mg / kg followed by 20 mg / kg body weight /day in two divided dose for 1 week and then in three divided dose up to 1 month.
Schedule of Vancomycin
H
Storage Requirements for Vancomycin
Store in room temperature. Keep away from moisture and light.
Effects of Missed Dosage of Vancomycin
Take the missed dose as soon as noticed and if it is the time for next dose then skip the missed dose. Continue the regular schedule. Do not double the dose.
Effects of Overdose of Vancomycin
Give supportive treatment and measures. Maintain glomerular filtration rate. Then if needed haemodialysis or haemoperfusion can be done.

Home Delivery for Ceftriaxone + Vancomycin in Your City

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However, we do publish a comprehensive directory of Pharmacies, Chemists and Druggists in cities all over India. You can use this directory to find the medicine stores in your city (or area) that provide home delivery services for ceftriaxone + vancomycin and other medicines and health products. Home delivery services for ceftriaxone + vancomycin may be free or they may cost you depending on the pharmacy and the minimum order requirements. It would be best to get this clarified while placing the order.

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Ceftriaxone + Vancomycin is a generic medicine name and there are several brands available for it. Some of the brands for ceftriaxone + vancomycin might be better known than ceftriaxone + vancomycin itself. If the pharmacy that's willing to deliver medicines to your home doesn't have ceftriaxone + vancomycin in stock, you can ask for one of the branded alternatives for ceftriaxone + vancomycin.