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- Pharmacology For Mosapride + Simethicone
Mosapride + Simethicone Pharmacology
Mosapride + Simethicone
About Mosapride + SimethiconeN/AMechanism of Action of Mosapride + SimethiconeN/APharmacokinets of Mosapride + SimethiconeN/AOnset of Action for Mosapride + SimethiconeN/ADuration of Action for Mosapride + SimethiconeN/AHalf Life of Mosapride + SimethiconeN/ASide Effects of Mosapride + SimethiconeN/AContra-indications of Mosapride + SimethiconeN/ASpecial Precautions while taking Mosapride + SimethiconeN/APregnancy Related InformationN/AOld Age Related InformationN/ABreast Feeding Related InformationN/AChildren Related InformationN/AIndications for Mosapride + SimethiconeN/AInteractions for Mosapride + SimethiconeN/ATypical Dosage for Mosapride + SimethiconeN/ASchedule of Mosapride + SimethiconeN/AStorage Requirements for Mosapride + SimethiconeN/AEffects of Missed Dosage of Mosapride + SimethiconeN/AEffects of Overdose of Mosapride + SimethiconeN/AMosapride
About MosaprideA selective 5HT4 agonist, A gastroprokinetic agent.Mechanism of Action of MosaprideMosapride is a Prokinetic drug. It is a 5 HT4 receptor agonist as well as 5HT3 receptor antagonist in the myenteric plexus. Enterochromaffin cells in the gastrointestinal mucosa produces and releases serotonin in response to stimuli (chemical or mechanical stimulation).Serotonin will enhances peristaltic movement by stimulating sensory neurons in the myenteric plexus. Stimulation of 5HT4 receptors will increase the release of Acetylcholine. The metabolite of Mosapride produces 5HT3 receptor antagonism and suppresses the inhibitory transmission in myenteric plexus. These all results in increased oesophageal peristaltic activity, lower oesophageal sphincter tone and enhances intestinal propulsive activity.Pharmacokinets of MosaprideAbsorption:It is absorbed after oral administration.Excretion: It is excreted mainly urine and faeces.
Onset of Action for MosaprideN/ADuration of Action for MosaprideN/AHalf Life of Mosapride2 - 3 hoursSide Effects of Mosapride1.Diarrhoea
2.Abdominal cramps
3.Headache
4.Dry mouth
5.Nausea
Contra-indications of Mosapride1.Hypersensitivity to MosaprideSpecial Precautions while taking Mosapride1.Hepatic impairment
2.Renal impairment
Pregnancy Related InformationUse with cautionOld Age Related InformationUse with cautionBreast Feeding Related InformationUse with cautionChildren Related InformationContraindicated
NEONATES: contraindicated
Indications for Mosapride1.Gastroesophageal reflux diseases
2.Functional dyspepsia
3.Diabetic gastropathy
4.Disorders associated with decreased gastric motility
5.Nausea
Interactions for MosaprideMosapride`s major degradation system is the cytochrome P450 (3A4) system. However, electrophysiological studies show that coadministration of drugs that inhibit the CYP 3A4 enzymes (erythromycin, ketoconazole, fluconazole, etc.) have no effect on mosapride indicating that a satisfactory safety margin exists in relation to rhythm abnormalities, unlike that which occurs with cisapride. Typical Dosage for MosaprideAdult:
Oral:2.5 - 10 mg every 6 - 8 hours in a day with meals
Children:not recommended
Schedule of MosaprideN/AStorage Requirements for MosaprideStore at 15 - 30 degree C in a tightly closed container. Protect from heat and light. Keep out of the reach of childrenEffects of Missed Dosage of MosaprideTake the missed dose as soon as noticed and if it is the time for next dose then skip the missed dose. Continue the regular schedule. Do not double the dose.
Effects of Overdose of MosaprideGive supportive measures and symptomatic treatment.
Simethicone
About SimethiconeOral anti-foaming agent, Silicones, Antiflatulent.Mechanism of Action of SimethiconeThis anti-gas (anti-flatulence) medication acts in the stomach and intestines to change the surface tension of gas bubbles, enabling smaller bubbles to join together into bigger bubbles. It results elimination of gas more easily by belching or passing flatus.Pharmacokinets of SimethiconeExcretion- Excreted through feces.Onset of Action for SimethiconeN/ADuration of Action for SimethiconeN/AHalf Life of SimethiconeN/ASide Effects of Simethicone1. Bloating
2. Constipation
3. Diarrhea
4. Gas
5. Heartburn
Contra-indications of Simethicone1. Hypersensitivity to the drug
2. Liver disease
3. Kidney disease
4. Serious illness
Special Precautions while taking Simethicone1.Swallow the tablets and capsules with a full glass of water.
2.Chew the chewable tablets thoroughly before swallowing.
3.Shake the drops well before using them.
4.To make administration easier, the drops can be mixed with 30 ml (2 tablespoons) of water or another liquid.
Pregnancy Related InformationUse with cautionOld Age Related InformationUse with cautionBreast Feeding Related InformationUse with cautionChildren Related InformationUse with cautionIndications for Simethicone1. Abdominal pain which is due to excessive gas in the digestive tract
2. Before gastroscopy or radiography of the bowel
Interactions for SimethiconeN/ATypical Dosage for SimethiconeOral-
Adults and teenagers-
60 -125mg four times a day, after meals and at bedtime. Not more than 500 mg should be taken in twenty-four hours.
Chewable tablets:
Adults and teenagers-
40 -125 mg four times a day, after meals and at bedtime or 150 mg three times a day, after meals. Not more than 500 mg should be taken in twenty-four hours.
Suspension:
Adults and teenagers-
40 -95 mg four times a day, after meals and at bedtime. Not more than 500 mg should be taken in twenty-four hours.
Schedule of SimethiconeN/AStorage Requirements for SimethiconeStored at room temperature (15-30?C) away from moisture and heat.Effects of Missed Dosage of SimethiconeTake the missed dose as soon as noticed and if it is the time for next dose then skip the missed dose. Continue the regular schedule. Do not double the dose.Effects of Overdose of SimethiconeGive symptomatic and supportive treatment.Home Delivery for Mosapride + Simethicone in Your City
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Mosapride + Simethicone is a generic medicine name and there are several brands available for it. Some of the brands for mosapride + simethicone might be better known than mosapride + simethicone itself. If the pharmacy that's willing to deliver medicines to your home doesn't have mosapride + simethicone in stock, you can ask for one of the branded alternatives for mosapride + simethicone.